| Substrate | A9273, Ala-Ala-Val-Ala p-nitroanilide |
| | S8758, N-Succinyl-Ala-Ala-Phe-7-amido-4-methylcoumarin |
| | S7388, N-Succinyl-Ala-Ala-Pro-Phe p-nitroanilide |
| | M4507, 4-Methylumbelliferyl p-trimethylammoniocinnamate chloride |
| | S9761, N-Succinyl-Ala-Ala-Pro-Phe-7-amido-4-methylcoumarin |
| | G3769, Glutaryl-Ala-Ala-Phe-4-methoxy-β-naphthylamide |
| | S1899, N-Succinyl-Gly-Gly-Phe-p-nitroanilide |
| | A3401, Ala-Ala-Phe-7-amido-4-methylcoumarin |
| | G4636, N-Glutaryl-Gly-Gly-Phe-β-naphthylamide |
| Inhibitor | A9285, α1-Antichymotrypsin from human plasma |
| | D0879, Diisopropylfluorophosphate |
| | A1153, Aprotinin from bovine lung |
| | A2504, 6-Aminocaproic acid |
| | T1886, Trypsin inhibitor from chicken egg white |
| | E1398, Ecotin |
| | T9777, Trypsin-chymotrypsin inhibitor from Glycine max (soybean) |
| | T4376, N-p-Tosyl-L-phenylalanine chloromethyl ketone |
| | B1552, Bromoenol lactone |
| | P7626, Phenylmethanesulfonyl fluoride |
| | A9024, α1-Antitrypsin from human plasma |
| | E7888, N-Acetyl-eglin C |
| | L2023, Leupeptin trifluoroacetate salt |
| | A6150, α1-Antitrypsin from human plasma |
| | A7824, 6-Aminocaproic acid |
| | C7268, Chymostatin |